Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3153 (2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4-hydroxybenzen...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3252 ((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3152 (2-{[2,6-dihydroxy-4-({[(3R,4R)-4-[(4-hydroxybenzen...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3248 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3243 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 18 | n/a | n/a | n/a | n/a | 7.5 | 30 |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3249 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3250 (2-[(4-hydroxybenzene)amido]cyclopentyl 3,5-dihydro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3149 (2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | Article | n/a | n/a | 32 | n/a | n/a | n/a | n/a | 7.5 | 30 |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3254 ((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3244 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 50 | n/a | n/a | n/a | n/a | 7.5 | 30 |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3253 ((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 67 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3245 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 80 | n/a | n/a | n/a | n/a | 7.5 | 30 |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3246 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3251 ((1S,2S)-2-[(4-hydroxybenzene)amido]cyclopentyl 3,5...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C delta type (Homo sapiens (Human)) | BDBM3247 ((3R,4R)-4-[(4-hydroxybenzene)amido]pyrrolidin-3-yl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
Sphinx Pharmaceuticals | Assay Description The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his... | Bioorg Med Chem Lett 5: 2133-8 (1995) Article DOI: 10.1016/0960-894X(95)00361-V BindingDB Entry DOI: 10.7270/Q26T0JT4 | |||||||||||
More data for this Ligand-Target Pair |